51458 Results for: "CAYMAN"

Atipamezole is an imidazole that potently antagonizes the 2-adrenoceptor (Ki = 1.6 nM).{25705,25706} It shows selectivity over the 1-adrenoceptor (Ki = 13,300 nM) and is a poor antagonist at a wide variety of other receptors and channels.{25706} Th 1 * 5 mg

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L-165,041 is a potent and selective agonist of the nuclear receptor PPAR/ (Ki = 9 nM, EC50 = 500 nM for hPPAR/).{7166,10670} It is less effective against PPAR and PPAR, with activity at those receptors depending on cell type and system of stu 1 * 25 mg

Supplier: CAYMAN

L-165,041 is a potent and selective agonist of the nuclear receptor PPAR/ (Ki = 9 nM, EC50 = 500 nM for hPPAR/).{7166,10670} It is less effective against PPAR and PPAR, with activity at those receptors depending on cell type and system of stu 1 * 25 mg

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L-165,041 is a potent and selective agonist of the nuclear receptor PPAR/ (Ki = 9 nM, EC50 = 500 nM for hPPAR/).{7166,10670} It is less effective against PPAR and PPAR, with activity at those receptors depending on cell type and system of stu 1 * 10 mg

Supplier: CAYMAN

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Yangonin is a natural kavalactone from the kava plant, P. methysticum. It enhances the binding of bicuculline at the γ-amino butyric acid (GABA) receptor GABAA at 1.0 µM.{25728} Yangonin also binds the central cannabinoid (CB1) receptor with a Ki va 1 * 5 mg

Supplier: CAYMAN

Yangonin is a natural kavalactone from the kava plant, P. methysticum. It enhances the binding of bicuculline at the γ-amino butyric acid (GABA) receptor GABAA at 1.0 µM.{25728} Yangonin also binds the central cannabinoid (CB1) receptor with a Ki va 1 * 5 mg

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Rauwolscine is a natural alkaloid that acts as a selective and reversible 2-adregenergic receptor antagonist (Ki = 12 nM).{25653} I t is a stereoisomer of yohimbine, which potently antagonizes both 1- and 2-adrenergic receptors.{25653} Rauwolscine 1 * 250 mg

Supplier: CAYMAN

Rauwolscine is a natural alkaloid that acts as a selective and reversible 2-adregenergic receptor antagonist (Ki = 12 nM).{25653} I t is a stereoisomer of yohimbine, which potently antagonizes both 1- and 2-adrenergic receptors.{25653} Rauwolscine 1 * 250 mg

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6-Thioguanine (6-TG) is a thio analog of the purine base guanine that incorporates into DNA during replication, inducing double-stra nd breaks that destabilize its structure and result in cytotoxicity.{25754,25756} Upon incorporation into DNA, 6-TG h 1 * 500 mg

Supplier: CAYMAN

6-Thioguanine (6-TG) is a thio analog of the purine base guanine that incorporates into DNA during replication, inducing double-stra nd breaks that destabilize its structure and result in cytotoxicity.{25754,25756} Upon incorporation into DNA, 6-TG h 1 * 500 mg