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Protein kinase C (20-28) (myristoylated)
Protein kinase C (20-28) (myristoylated)
  ENZOBMLP2050500
 :  
Protein kinase C (20-28) (myristoylated)
  ENZOBMLP2050500
 :  

 

  • Förp.:
    0,5 mg
  • Seq:
    02
  • Protein/peptide name:
    Protein kinase C (20-28) (myristoylated)
  • Renhet:
    >98% (HPLC)
  • Formulering:
    TFA salt. Lyophilised.

 

 

PKC inhibitor

Pseudosubstrate sequence from PKCalpha and ß. Highly specific inhibitor, which is N-terminal myristoylated to allow membrane permeability. IC50=8 µM for TPA activation of MARCKS phosphorylation in fibroblast primary cultures, and 98% inhibition at 100 µM. Partially reverses multidrug resistance in human breast cancer cells.