22289 Results for: "3-(Trifluoromethoxy)pyrrolidine+hydrochloride"

Supplier: Cayman Chemical

A potent, cell-permeable inhibitor of SET7/9 (IC50 = 2 nM) that demonstrates greater than 1,000-fold selectivity over a panel of 18 other methyltransferases 1 * 5 mg

Supplier: Cayman Chemical

A slow, tight binding, competitive aminopeptidase (AP) inhibitor, first described as an inhibitor of AP-A (glutamyl AP 1 * 5 mg

Supplier: Cayman Chemical

A dual orexin 1 and 2 receptor antagonist (Kds = 1.3 and 0.17 nM, respectively) 1 * 10 mg

Supplier: Apollo Scientific

BMS_582949 hydrochloride_25mg pack 1 * 25 mg

Supplier: Apollo Scientific

Ulixertinib hydrochloride_50mg pack 1 * 50 mg

Supplier: Apollo Scientific

GDC_0994 hydrochloride_5mg pack 1 * 5 mg

Supplier: Cayman Chemical

A fluoroquinolone antibiotic that displays broad spectrum antibacterial activity by inhibiting the bacterial regulatory enzyme DNA g yrase (IC50 = 0.92 µg/ml) as well as topoisomerase IV (IC50 = 1.62 µg/ml) 1 * 250 mg

Supplier: Cayman Chemical

A β1 adrenergic receptor antagonist and a β2 adrenergic receptor partial agonist that relaxes human arteries and veins with ED50 val ues of 40-50 µM in vitro 1 * 1 mg

Supplier: Cayman Chemical

A β1 adrenergic receptor antagonist and a β2 adrenergic receptor partial agonist that relaxes human arteries and veins with ED50 val ues of 40-50 µM in vitro 1 * 5 mg

Supplier: Cayman Chemical

A prodrug of benazeprilat inhibits enzymatic activity of partially purified ACE isolated from rabbit lung (IC50 = 2 nM) 1 * 50 mg

Supplier: Cayman Chemical

An active metabolite of proguanil, produced by CYP2C19 1 * 25 mg

Supplier: Cayman Chemical

A potent inhibitor of MELK (IC50 = 0.41 nM) 1 * 1 mg

Supplier: Cayman Chemical

A potent inhibitor of JAK2 that also inhibits the JAK2V617F mutant enzyme (IC50s for both enzymes 0.5 nM) 1 * 5 mg

Supplier: Cayman Chemical

A steroidal alkaloid that suppresses NF-B signaling in LPS-stimulated macrophages, blocking induced expression of iNOS and COX-2 1 * 50 mg

Supplier: Cayman Chemical

An inhibitor of JAK3 (IC50 = 79 nM) 1 * 5 mg

Supplier: Cayman Chemical

A broad-spectrum, indole-based antiviral compound that blocks viral fusion with target membranes, prohibiting viral entry into cells 1 * 100 mg

Supplier: Apollo Scientific

LY2584702 Hydrochloride_50mg pack 1 * 50 mg

Supplier: Apollo Scientific

SB_203580 Hydrochloride_50mg pack 1 * 50 mg

Supplier: Cayman Chemical

A selective, reversible inhibitor of MAO-B (Ki = 0.091 M) over MAO-A (Ki = 9.06 M) 1 * 100 mg

Supplier: Cayman Chemical

A cell-permeable inhibitor of Hhat (IC50 = 0.85 µM) 1 * 5 mg

Supplier: Cayman Chemical

1-2-(4-methoxyphenyl)-2-3-(4-methoxyphenyl)propoxyethyl-1H-i midazole,monohydrochloride 1 * 5 mg

Supplier: Cayman Chemical

A selective antagonist of GABAB receptors (IC50 = 43 µM) 1 * 1 mg

Supplier: Cayman Chemical

A potent inhibitor of MELK (IC50 = 0.41 nM) 1 * 10 mg

Supplier: Cayman Chemical

A conventional antipsychotic drug that potently activates several neuroreceptors, including serotonin (Kis = 10, 60, and 57 nM for 5 -HT2A, 5-HT2C, and 5-HT6, respectively), dopamine D2 (Ki = 11 nM), and adrenergic 1A (Ki = 5 nM) receptors 1 * 25 g

Supplier: Cayman Chemical

A fluoroquinolone antibiotic that displays broad spectrum antibacterial activity by inhibiting the bacterial regulatory enzyme DNA g yrase (IC50 = 0.92 µg/ml) as well as topoisomerase IV (IC50 = 1.62 µg/ml) 1 * 100 mg

Supplier: Cayman Chemical

A conventional antipsychotic drug that potently activates several neuroreceptors, including serotonin (Kis = 10, 60, and 57 nM for 5 -HT2A, 5-HT2C, and 5-HT6, respectively), dopamine D2 (Ki = 11 nM), and adrenergic 1A (Ki = 5 nM) receptors 1 * 1 g

Supplier: Cayman Chemical

A conventional antipsychotic drug that potently activates several neuroreceptors, including serotonin (Kis = 10, 60, and 57 nM for 5 -HT2A, 5-HT2C, and 5-HT6, respectively), dopamine D2 (Ki = 11 nM), and adrenergic 1A (Ki = 5 nM) receptors 1 * 5 g

Supplier: Cayman Chemical

A potent inhibitor of JAK2 that also inhibits the JAK2V617F mutant enzyme (IC50s for both enzymes 0.5 nM) 1 * 1 mg

Supplier: Cayman Chemical

2-3-(2,3-dichlorophenoxy)propylamino-ethanol, monohydrochloride 1 * 50 mg

Supplier: Cayman Chemical

A gastroprotective histamine H2 receptor antagonist (pKi = 7.1) that decreases gastric acid secretion and inhibits intracellular cAM P production (IC50 = 1 µM) 1 * 1 g