18721 Results for: "Neocuproine+hydrochloride+monohydrate"

Supplier: Cayman Chemical

A cell-permeable inhibitor of Hhat (IC50 = 0.85 µM) 1 * 1 mg

Supplier: Cayman Chemical

A pan inhibitor PKD (IC50s = 1, 2.5, and 2 nM for PKD1, PKD2, and PKD3, respectively) 1 * 10 mg

Supplier: Cayman Chemical

A major active metabolite of saxagliptin inhibits DPP-4 (Ki = 2.6 nM for human recombinant enzyme) 1 * 1 mg

Supplier: Cayman Chemical

A potent, selective antagonist of the serotonin (5-HT) receptor 5-HT3 (pKi = 10.4 in rat cortex) 1 * 10 mg

Supplier: Cayman Chemical

An active metabolite of proguanil, produced by CYP2C19 1 * 25 mg

Supplier: Cayman Chemical

A benzazepine derivative that antagonizes the binding of AVP to vasopressin V2 receptors (IC50 = 14 nM) 1 * 10 mg

Supplier: Cayman Chemical

A benzazepine derivative that antagonizes the binding of AVP to vasopressin V2 receptors (IC50 = 14 nM) 1 * 50 mg

Supplier: Cayman Chemical

A broad-spectrum, indole-based antiviral compound that blocks viral fusion with target membranes, prohibiting viral entry into cells 1 * 5 mg

Supplier: Cayman Chemical

A selective antagonist of GABAB receptors (IC50 = 43 µM) 1 * 10 mg

Supplier: Cayman Chemical

A potent, cell-permeable inhibitor of SET7/9 (IC50 = 2 nM) that demonstrates greater than 1,000-fold selectivity over a panel of 18 other methyltransferases 1 * 1 mg

Supplier: Apollo Scientific

LY2584702 Hydrochloride_50mg pack 1 * 50 mg

Supplier: Apollo Scientific

SB_203580 Hydrochloride_50mg pack 1 * 50 mg

Supplier: Cayman Chemical

A slow, tight binding, competitive aminopeptidase (AP) inhibitor, first described as an inhibitor of AP-A (glutamyl AP 1 * 500 µG

Supplier: Cayman Chemical

A fluoroquinolone antibiotic that displays broad spectrum antibacterial activity by inhibiting the bacterial regulatory enzyme DNA g yrase (IC50 = 0.92 µg/ml) as well as topoisomerase IV (IC50 = 1.62 µg/ml) 1 * 100 mg

Supplier: Cayman Chemical

A conventional antipsychotic drug that potently activates several neuroreceptors, including serotonin (Kis = 10, 60, and 57 nM for 5 -HT2A, 5-HT2C, and 5-HT6, respectively), dopamine D2 (Ki = 11 nM), and adrenergic 1A (Ki = 5 nM) receptors 1 * 25 g

Supplier: Apollo Scientific

GDC_0994 hydrochloride_1mg pack 1 * 1 mg

Supplier: Cayman Chemical

A broad-spectrum, indole-based antiviral compound that blocks viral fusion with target membranes, prohibiting viral entry into cells 1 * 10 mg

Supplier: Cayman Chemical

A selective, reversible inhibitor of MAO-B (Ki = 0.091 M) over MAO-A (Ki = 9.06 M) 1 * 100 mg

Supplier: Cayman Chemical

A cell-permeable inhibitor of Hhat (IC50 = 0.85 µM) 1 * 5 mg

Supplier: Cayman Chemical

A blocker of KCNQ channels that potently inhibits KCNQ1 and 2 homomeric channels (IC50 = 0.75 and 0.71 µM, respectively) as well as KCNQ2+3 heteromultimers (IC50 = 0.6 µM) 1 * 5 mg

Supplier: Cayman Chemical

An ATP-competitive, pan-Akt kinase inhibitor (IC50s = 2, 13, and 9 nM for Akt1, 2, and 3, respectively) that inhibits proliferation and induces apoptosis in various human tumor cells in vitro and in xenografts in immunocompromised mice 1 * 5 mg

Supplier: Cayman Chemical

A potent inhibitor of JAK2 that also inhibits the JAK2V617F mutant enzyme (IC50s for both enzymes 0.5 nM) 1 * 10 mg

Supplier: Cayman Chemical

A potent inhibitor of IB kinases (IKKs), displaying IC50 values of 200, 40, and 70 nM for IKK, IKK, and IKK complex, respectively , in cell-free assays 1 * 5 mg

Supplier: Cayman Chemical

A potent inhibitor of JAK2 that also inhibits the JAK2V617F mutant enzyme (IC50s for both enzymes 0.5 nM) 1 * 1 mg

Supplier: Apollo Scientific

BMS_582949 hydrochloride_5mg pack 1 * 5 mg

Supplier: Cayman Chemical

An inhibitor of JAK3 (IC50 = 79 nM) 1 * 1 mg

Supplier: Apollo Scientific

LY2584702 Hydrochloride_25mg pack 1 * 25 mg

Supplier: Apollo Scientific

SB_203580 Hydrochloride_10mg pack 1 * 10 mg

Supplier: Cayman Chemical

An antibiotic that can inhibit cell wall synthesis in plant-pathogenic oomycetes (MIC = 25 µg/ml for P. medicaginis M2913) and certa in fungi as well as some bacterial species (MIC = 400 µg/ml for S. aureus) 1 * 5 mg

Supplier: Cayman Chemical

An ATP-competitive, pan-Akt kinase inhibitor (IC50s = 2, 13, and 9 nM for Akt1, 2, and 3, respectively) that inhibits proliferation and induces apoptosis in various human tumor cells in vitro and in xenografts in immunocompromised mice 1 * 10 mg