17599 Results for: "Cyclopropanecarboxamidine+hydrochloride"

Supplier: Cayman Chemical

A potent inhibitor of MELK (IC50 = 0.41 nM) 1 * 5 mg

Supplier: Cayman Chemical

A fluoroquinolone antibiotic that displays broad spectrum antibacterial activity by inhibiting the bacterial regulatory enzyme DNA g yrase (IC50 = 0.92 µg/ml) as well as topoisomerase IV (IC50 = 1.62 µg/ml) 1 * 250 mg

Supplier: Apollo Scientific

SB_203580 Hydrochloride_50mg pack 1 * 50 mg

Supplier: Apollo Scientific

LY2584702 Hydrochloride_50mg pack 1 * 50 mg

Supplier: Cayman Chemical

An orally active, selective inhibitor of Cdk4 (IC50 = 11 nM) and Cdk6 (IC50 = 16 nM) with antiproliferative activity against retinob lastoma-positive tumor cells, blocking retinoblastoma phosphorylation and inducing G1 arrest 1 * 1 mg

Supplier: Cayman Chemical

An antibiotic that can inhibit cell wall synthesis in plant-pathogenic oomycetes (MIC = 25 µg/ml for P. medicaginis M2913) and certa in fungi as well as some bacterial species (MIC = 400 µg/ml for S. aureus) 1 * 25 mg

Supplier: Cayman Chemical

A cell-permeable inhibitor of Hhat (IC50 = 0.85 µM) 1 * 1 mg

Supplier: Cayman Chemical

1-2-(4-methoxyphenyl)-2-3-(4-methoxyphenyl)propoxyethyl-1H-i midazole,monohydrochloride 1 * 10 mg

Supplier: Cayman Chemical

A -adrenergic receptor agonist with potent positive inotropic effects in vivo 1 * 5 mg

Supplier: Cayman Chemical

A dual orexin 1 and 2 receptor antagonist (Kds = 1.3 and 0.17 nM, respectively) 1 * 5 mg

Supplier: Cayman Chemical

Selectively inhibits human NHE-1 with an IC50 value of 14 nM 1 * 1 mg

Supplier: Cayman Chemical

Selectively inhibits human NHE-1 with an IC50 value of 14 nM 1 * 5 mg

Supplier: Cayman Chemical

1R,2,3,4,4aS,9,10,10aR-octahydro-1,4a-dimethyl-7-(1-methylethyl) -1-phenanthrenemethanamine, monohydrochloride 1 * 5 mg

Supplier: Cayman Chemical

A conventional antipsychotic drug that potently activates several neuroreceptors, including serotonin (Kis = 10, 60, and 57 nM for 5 -HT2A, 5-HT2C, and 5-HT6, respectively), dopamine D2 (Ki = 11 nM), and adrenergic 1A (Ki = 5 nM) receptors 1 * 25 g

Supplier: Cayman Chemical

A fluoroquinolone antibiotic that displays broad spectrum antibacterial activity by inhibiting the bacterial regulatory enzyme DNA g yrase (IC50 = 0.92 µg/ml) as well as topoisomerase IV (IC50 = 1.62 µg/ml) 1 * 100 mg

Supplier: Cayman Chemical

A first generation tricyclic antidepressant 1 * 5 g

Supplier: Cayman Chemical

A potent, cell-permeable inhibitor of SET7/9 (IC50 = 2 nM) that demonstrates greater than 1,000-fold selectivity over a panel of 18 other methyltransferases 1 * 1 mg

Supplier: Cayman Chemical

A benzazepine derivative that antagonizes the binding of AVP to vasopressin V2 receptors (IC50 = 14 nM) 1 * 5 mg

Supplier: Cayman Chemical

An active metabolite of proguanil, produced by CYP2C19 1 * 50 mg

Supplier: Cayman Chemical

1-2-(4-methoxyphenyl)-2-3-(4-methoxyphenyl)propoxyethyl-1H-i midazole,monohydrochloride 1 * 1 mg

Supplier: Cayman Chemical

A dual orexin 1 and 2 receptor antagonist (Kds = 1.3 and 0.17 nM, respectively) 1 * 10 mg

Supplier: Cayman Chemical

A slow, tight binding, competitive aminopeptidase (AP) inhibitor, first described as an inhibitor of AP-A (glutamyl AP 1 * 5 mg

Supplier: Cayman Chemical

A blocker of KCNQ channels that potently inhibits KCNQ1 and 2 homomeric channels (IC50 = 0.75 and 0.71 µM, respectively) as well as KCNQ2+3 heteromultimers (IC50 = 0.6 µM) 1 * 5 mg

Supplier: Cayman Chemical

An epimer of chlortetracycline 1 * 1 mg

Supplier: Cayman Chemical

A steroidal alkaloid that suppresses NF-B signaling in LPS-stimulated macrophages, blocking induced expression of iNOS and COX-2 1 * 50 mg

Supplier: Cayman Chemical

A potent inhibitor of JAK2 that also inhibits the JAK2V617F mutant enzyme (IC50s for both enzymes 0.5 nM) 1 * 5 mg

Supplier: Apollo Scientific

LY2584702 Hydrochloride_25mg pack 1 * 25 mg

Supplier: Cayman Chemical

An orally active, selective inhibitor of Cdk4 (IC50 = 11 nM) and Cdk6 (IC50 = 16 nM) with antiproliferative activity against retinob lastoma-positive tumor cells, blocking retinoblastoma phosphorylation and inducing G1 arrest 1 * 25 mg

Supplier: Cayman Chemical

A dual orexin 1 and 2 receptor antagonist (Kds = 1.3 and 0.17 nM, respectively) 1 * 1 mg

Supplier: Cayman Chemical

An ATP-competitive, pan-Akt kinase inhibitor (IC50s = 2, 13, and 9 nM for Akt1, 2, and 3, respectively) that inhibits proliferation and induces apoptosis in various human tumor cells in vitro and in xenografts in immunocompromised mice 1 * 10 mg