K-252b ≥98% (by HPLC)
General, cell permeable protein kinase inhibitor. Acts by binding to the ATP binding domain of the kinase. Potent inhibitor of Ca2+/calmodulin kinase II. Inhibits myosin light chain kinase (MLCK; Ki=0.147µM), cAMP- dependent protein kinase (PKA; Ki=0.09µM), protein kinase C (PKC; Ki=0.02µM), and cGMP-dependent protein kinase (PKG; Ki=0.1µM).
- PKC inhibitor
White solid.
Soluble in DMSO (1mg/ml) or dimethyl formamide (1mg/ml).
- :99570-78-2
- :C₂₆H₁₉N₃O₅
- :453.5 g/mol
- :Refrigerator
- Pk:100 µG
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