"MEDCHEMEXPRESS"
SOLUBILITY: DISSOLVE IN DMSO
PENTAGASTRIN IS A SYNTHETIC POLYPEPTIDE THAT HAS EFFECTS LIKE GASTRIN WHEN GIVEN PARENTERALLY,WHICH CAN CAUSE THE SECRETION AND SYNTHESIS OF SALIVARY PROTEINS.[1]IN VIVO: WIN55, 212-2, WHICH IS A NON-SELECTIVE CANNABIN 1 * 10 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: DISSOLVE IN DMSO
PENTAGASTRIN IS A SYNTHETIC POLYPEPTIDE THAT HAS EFFECTS LIKE GASTRIN WHEN GIVEN PARENTERALLY,WHICH CAN CAUSE THE SECRETION AND SYNTHESIS OF SALIVARY PROTEINS.[1]IN VIVO: WIN55, 212-2, WHICH IS A NON-SELECTIVE CANNABIN 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO > 45 MG/ML WATER < 1 MG/ML
RG7388 IS AN ORAL, SELECTIVE, SMALL MOLECULE MD M2 ANTAGONIST THAT INHIBITS BINDING OF MDM2 TO P53. IC50 VALUE: 30 NM (AVERAGE IC50 OF THREE WT-P53 CANCER CELL LINES 1 * 100 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO > 45 MG/ML WATER < 1 MG/ML
RG7388 IS AN ORAL, SELECTIVE, SMALL MOLECULE MD M2 ANTAGONIST THAT INHIBITS BINDING OF MDM2 TO P53. IC50 VALUE: 30 NM (AVERAGE IC50 OF THREE WT-P53 CANCER CELL LINES 1 * 100 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 100 MM IN DMSO;
FR180204 IS A POTENT AND SELECTIVE ATP-COMPETITIVE INHIBITOR OF ERK1 AND ERK2 WITH KI VALUE OF 0.31 UM AND 0.14 UM RESPECTIVELY HAS IC50 VALUES OF 0.51 AND 0.33 ΜM IN ENZYMATIC ASSA 1 * 1 mL
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 100 MM IN DMSO;
FR180204 IS A POTENT AND SELECTIVE ATP-COMPETITIVE INHIBITOR OF ERK1 AND ERK2 WITH KI VALUE OF 0.31 UM AND 0.14 UM RESPECTIVELY HAS IC50 VALUES OF 0.51 AND 0.33 ΜM IN ENZYMATIC ASSA 1 * 1 mL
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SOLUBILITY: 10 MM IN DMSO
ENDOXIFEN IS THE MOST IMPORTANT TAMOXIFEN METABOLITE RESPONSIBLE FOR ELICITING THE ANTI-ESTROGENIC EFFE CTS OF THIS DRUG IN BREAST CANCER CELLS EXPRESSING ESTROGEN RECEPTOR-ALPHA (ERΑ). ENDOXIFEN INHIBITS HERG TAIL CURREN 1 * 5 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: 10 MM IN DMSO
ENDOXIFEN IS THE MOST IMPORTANT TAMOXIFEN METABOLITE RESPONSIBLE FOR ELICITING THE ANTI-ESTROGENIC EFFE CTS OF THIS DRUG IN BREAST CANCER CELLS EXPRESSING ESTROGEN RECEPTOR-ALPHA (ERΑ). ENDOXIFEN INHIBITS HERG TAIL CURREN 1 * 5 mg
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SOLUBILITY: 10 MM IN DMSO
TRIMIPRAMINE MALEATE IS A SEROTONIN TRANSPORT AND NOREPINEPHRINE UPTAKE BLOCKER, IS A TRICYCLIC ANTIDEP RESSANT (TCA) WITH ANTIPSYCHOTIC AND SEDATIVE PROPERTIES. 1 * 100 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: 10 MM IN DMSO
TRIMIPRAMINE MALEATE IS A SEROTONIN TRANSPORT AND NOREPINEPHRINE UPTAKE BLOCKER, IS A TRICYCLIC ANTIDEP RESSANT (TCA) WITH ANTIPSYCHOTIC AND SEDATIVE PROPERTIES. 1 * 100 mg
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STING agonist-4 ,98% 1 * 10 mg
Supplier: MEDCHEMEXPRESS
STING agonist-4 ,98% 1 * 10 mg
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CCT251236 10 mM 1 mL IN DMSO 1 * 1 mL
Supplier: MEDCHEMEXPRESS
CCT251236 10 mM 1 mL IN DMSO 1 * 1 mL
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 90 MG/ML WATER <1 MG/ML
DOFETILIDE(TIKOSYN) IS A CLASS III ANTIARRHYTHMIC AGENT.TARGET: POTASSIUM CHANNELIN PATIENTS WITH CONGESTIVE HEART FAILURE AND REDUCED LEFT VENTRICULAR FUNCTION, DOFETI 1 * 50 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 90 MG/ML WATER <1 MG/ML
DOFETILIDE(TIKOSYN) IS A CLASS III ANTIARRHYTHMIC AGENT.TARGET: POTASSIUM CHANNELIN PATIENTS WITH CONGESTIVE HEART FAILURE AND REDUCED LEFT VENTRICULAR FUNCTION, DOFETI 1 * 50 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: > 5.1 MG/ML, H2O: < 1 MG/ML
CHIR-99021 (CT99021) IS A GSK-3Α/Β INHIBITOR W ITH IC50 OF 10 NM/6.7 NM > 500-FOLD SELECTIVITY FOR GSK-3 VERSUS ITS CLOSEST HOMOLOGS CDC2 AND ERK2, AS WELL AS OTHE 1 * 50 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: > 5.1 MG/ML, H2O: < 1 MG/ML
CHIR-99021 (CT99021) IS A GSK-3Α/Β INHIBITOR W ITH IC50 OF 10 NM/6.7 NM > 500-FOLD SELECTIVITY FOR GSK-3 VERSUS ITS CLOSEST HOMOLOGS CDC2 AND ERK2, AS WELL AS OTHE 1 * 50 mg
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SOLUBILITY: H2O (100 MM) OR PBS (100 MM)
Y-27632 IS A SELECTIVE ROCK1 (P160ROCK) INHIBITOR WITH KI OF 140 NM, EXHIBITS >200-FOLD SELECTIVITY OVER OTHER KINASES, INCLUDING PKC, CAMP-DEPENDENT PROTEIN KINASE, MLCK AND PAK.IC50 VALUE: 140 NM (KI)TARG 1 * 5 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: H2O (100 MM) OR PBS (100 MM)
Y-27632 IS A SELECTIVE ROCK1 (P160ROCK) INHIBITOR WITH KI OF 140 NM, EXHIBITS >200-FOLD SELECTIVITY OVER OTHER KINASES, INCLUDING PKC, CAMP-DEPENDENT PROTEIN KINASE, MLCK AND PAK.IC50 VALUE: 140 NM (KI)TARG 1 * 5 mg
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Luxdegalutamide-98% 1 * 10 mg
Supplier: MEDCHEMEXPRESS
Luxdegalutamide-98% 1 * 10 mg



