"MEDCHEMEXPRESS"
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
MI-773 IS AN ORALLY AVAILABLE SPIRO-OXINDOLE HDM2 (HUMAN DOUBLE MI NUTE 2) ANTAGONIST WITH POTENTIAL ANTINEOPLASTIC ACTIVITY.IC50 VALUE:TARGET: HDM2-P53UPON ORAL ADMINISTRATION, THE P5 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
MI-773 IS AN ORALLY AVAILABLE SPIRO-OXINDOLE HDM2 (HUMAN DOUBLE MI NUTE 2) ANTAGONIST WITH POTENTIAL ANTINEOPLASTIC ACTIVITY.IC50 VALUE:TARGET: HDM2-P53UPON ORAL ADMINISTRATION, THE P5 1 * 10 mg
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DAGROCORAT HYDROCHLORIDE 1 * 5 mg
Supplier: MEDCHEMEXPRESS
DAGROCORAT HYDROCHLORIDE 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 75 MG/ML WATER <1 MG/ML ETHANOL <1 MG/ML
BMN 673 IS A NOVEL PARP1/2 INHIB ITOR WITH IC50 OF 0.58 NM(PARP1) DOES NOT INHIBIT PARG AND IS HIGHLY SENSITIVE TO PTEN MUTATION. IC50 VALUE: 0.58 NM 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 75 MG/ML WATER <1 MG/ML ETHANOL <1 MG/ML
BMN 673 IS A NOVEL PARP1/2 INHIB ITOR WITH IC50 OF 0.58 NM(PARP1) DOES NOT INHIBIT PARG AND IS HIGHLY SENSITIVE TO PTEN MUTATION. IC50 VALUE: 0.58 NM 1 * 10 mg
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SOLUBILITY: DMSO ≥45MG/ML WATER <1.2MG/ML ETHANOL <1.2.MG/ML
VELIPARIB (ABT-888) IS A POTENT INHIBITOR OF PARP1 AND PARP2 WITH KI OF 5.2 NM AND 2.9 NM, RESPECTIVELY.IC50 VALUE: 5.2 NM(KI FOR PARP1) 2.9 NM(KI FOR PARP2) [1]TARGET: PARP1 PARP2IN I 1 * 50 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: DMSO ≥45MG/ML WATER <1.2MG/ML ETHANOL <1.2.MG/ML
VELIPARIB (ABT-888) IS A POTENT INHIBITOR OF PARP1 AND PARP2 WITH KI OF 5.2 NM AND 2.9 NM, RESPECTIVELY.IC50 VALUE: 5.2 NM(KI FOR PARP1) 2.9 NM(KI FOR PARP2) [1]TARGET: PARP1 PARP2IN I 1 * 50 mg
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FLAVOPIRIDOL 10 MM * 1 ML IN DMSO 1 * 1 mL
Supplier: MEDCHEMEXPRESS
FLAVOPIRIDOL 10 MM * 1 ML IN DMSO 1 * 1 mL
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: 31MG/ML
A-1155463 IS A HIGHLY POTENT AND SELECTIVE BCL-XL INHIBITOR, A-115 5463 SHOWS PICOMOLAR BINDING AFFINITY TO BCL-XL (KI <0.01 NM), AND >1000-FOLD WEAKER BINDING TO BCL-2 (KI = 80 NM) AN 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: 31MG/ML
A-1155463 IS A HIGHLY POTENT AND SELECTIVE BCL-XL INHIBITOR, A-115 5463 SHOWS PICOMOLAR BINDING AFFINITY TO BCL-XL (KI <0.01 NM), AND >1000-FOLD WEAKER BINDING TO BCL-2 (KI = 80 NM) AN 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: 9 MG/ML, H2O: < 1 MG/ML
CRIZOTINIB (PF-2341066) IS A POTENT INHIBITOR OF C -MET AND ALK WITH IC50 OF 11 NM AND 24 NM, RESPECTIVLEY.IC50 VALUE: 11 NM/24 NM (C-MET/ALK) [1]TARGET: C-MET/ALKIN VI 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: 9 MG/ML, H2O: < 1 MG/ML
CRIZOTINIB (PF-2341066) IS A POTENT INHIBITOR OF C -MET AND ALK WITH IC50 OF 11 NM AND 24 NM, RESPECTIVLEY.IC50 VALUE: 11 NM/24 NM (C-MET/ALK) [1]TARGET: C-MET/ALKIN VI 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 52 MG/ML WATER <1 MG/ML
NECROSTATIN-1 IS A SPECIFIC RIP1 INHIBITOR AND INH IBITS TNF-Α-INDUCED NECROPTOSIS WITH EC50 OF 490 NM.IC50 VALUE: 490 NM (EC50)TARGET: TNF-ALPHANECROSTATIN-1 IS AN INH 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 52 MG/ML WATER <1 MG/ML
NECROSTATIN-1 IS A SPECIFIC RIP1 INHIBITOR AND INH IBITS TNF-Α-INDUCED NECROPTOSIS WITH EC50 OF 490 NM.IC50 VALUE: 490 NM (EC50)TARGET: TNF-ALPHANECROSTATIN-1 IS AN INH 1 * 10 mg
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Trastuzumab emtansine 1018448-65-1 1 * 5 mg
Supplier: MEDCHEMEXPRESS
Trastuzumab emtansine 1018448-65-1 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥78MG/ML WATER <1MG/ML ETHANOL ≥6MG/ML
ZM 336372 IS A POTENT AND SELECTIV E C-RAF INHIBITOR WITH IC50 OF 70 NM, 10-FOLD SELECTIVITY OVER B-RAF, NO INHIBITION TO PKA/B/C, AMPK, P70S6, ETC.IC50 1 * 1 mL
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥78MG/ML WATER <1MG/ML ETHANOL ≥6MG/ML
ZM 336372 IS A POTENT AND SELECTIV E C-RAF INHIBITOR WITH IC50 OF 70 NM, 10-FOLD SELECTIVITY OVER B-RAF, NO INHIBITION TO PKA/B/C, AMPK, P70S6, ETC.IC50 1 * 1 mL
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Xanthine-13C 15N2 (97%) 1mg 1 * 1 mg
Supplier: MEDCHEMEXPRESS
Xanthine-13C 15N2 (97%) 1mg 1 * 1 mg
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AA26-9 is a potent and broad spectrum serine hydrolase inhibitor. 1 * 5 mg
Supplier: MEDCHEMEXPRESS
AA26-9 is a potent and broad spectrum serine hydrolase inhibitor. 1 * 5 mg



