"MEDCHEMEXPRESS"
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
SAR7334 IS A NOVEL AND POTENT TRCP6 INHIBITOR FROM PCT INT. APPL. (2011), WO 2011107474 A1 20110909. 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
SAR7334 IS A NOVEL AND POTENT TRCP6 INHIBITOR FROM PCT INT. APPL. (2011), WO 2011107474 A1 20110909. 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: IN DMSO> 10 MM
RIMONABANT HCL(SR141716A) IS A SELECTIVE CENTRAL CANNABINOID (CB1 ) RECEPTOR INVERSE AGONIST WITH KI OF 1.8 NM.IC50 VALUE: 1.8 NM(KI)TARGET: CB1 RECEPTORIN VITRO: RIMONABANT DOSE-DEPE 1 * 100 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: IN DMSO> 10 MM
RIMONABANT HCL(SR141716A) IS A SELECTIVE CENTRAL CANNABINOID (CB1 ) RECEPTOR INVERSE AGONIST WITH KI OF 1.8 NM.IC50 VALUE: 1.8 NM(KI)TARGET: CB1 RECEPTORIN VITRO: RIMONABANT DOSE-DEPE 1 * 100 mg
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SOLUBILITY: DMSO ≥ 26 MG/ML
FCCP IS AN UNCOUPLER OF OXIDATIVE PHOSPHORYLATION IN MITOCHONDRIA. 1 * 10 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: DMSO ≥ 26 MG/ML
FCCP IS AN UNCOUPLER OF OXIDATIVE PHOSPHORYLATION IN MITOCHONDRIA. 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO >20 MG/ML
UK-5099(PF1005023) IS A POTENT INHIBITOR OF PLASMA MEMBRANE MONOC ARBOXYLATE TRANSPORTERS (MCTS) AND THE MITOCHONDRIAL PYRUVATE CARRIER (MPC) INHIBITS PYRUVATE-DEPENDENT O2 CONSUMPTI 1 * 1 mL
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO >20 MG/ML
UK-5099(PF1005023) IS A POTENT INHIBITOR OF PLASMA MEMBRANE MONOC ARBOXYLATE TRANSPORTERS (MCTS) AND THE MITOCHONDRIAL PYRUVATE CARRIER (MPC) INHIBITS PYRUVATE-DEPENDENT O2 CONSUMPTI 1 * 1 mL
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO (FREE SOLUBLE)
IRBINITINIB(ARRY-380 ONT-380) IS A POTENT AND SELE CTIVE HER2 INHIBITOR WITH IC50 OF 8 NM, EQUIPOTENT AGAINST TRUNCATED P95-HER2, 500-FOLD MORE SELECTIVE FOR HER2 VERSU 1 * 50 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO (FREE SOLUBLE)
IRBINITINIB(ARRY-380 ONT-380) IS A POTENT AND SELE CTIVE HER2 INHIBITOR WITH IC50 OF 8 NM, EQUIPOTENT AGAINST TRUNCATED P95-HER2, 500-FOLD MORE SELECTIVE FOR HER2 VERSU 1 * 50 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO:36MG/ML
AZD3965 IS A SELECTIVE INHIBITOR OF MONOCARBOXYLATE TRANSPORTER 1 ( MCT1) WITH A BINDING AFFINITY OF 1.6 NM, IS 6 FOLD SELECTIVE OVER MCT2 AND DOES NOT INHIBIT MCT4 AT 10 ΜM.IC50 VALUE: 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO:36MG/ML
AZD3965 IS A SELECTIVE INHIBITOR OF MONOCARBOXYLATE TRANSPORTER 1 ( MCT1) WITH A BINDING AFFINITY OF 1.6 NM, IS 6 FOLD SELECTIVE OVER MCT2 AND DOES NOT INHIBIT MCT4 AT 10 ΜM.IC50 VALUE: 1 * 5 mg
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SOLUBILITY: 10 MM IN DMSO
GLAFENINE IS A NON-STEROIDAL ANTI-INFLAMMATORY DRUG (NSAID), IS A NON-NARCOTIC ANALGESIC AGENT, WIDELY USED FOR THE TREATMENT OF PAINS OF VARIOUS ORIGINS. 1 * 100 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: 10 MM IN DMSO
GLAFENINE IS A NON-STEROIDAL ANTI-INFLAMMATORY DRUG (NSAID), IS A NON-NARCOTIC ANALGESIC AGENT, WIDELY USED FOR THE TREATMENT OF PAINS OF VARIOUS ORIGINS. 1 * 100 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 50 MG/ML
SCH772984 IS A NOVEL, SPECIFIC INHIBITOR OF ERK1/2 WITH IC50 OF 4 NM AND 1 NM, RESPECTIVELY.IC50 VALUE: 4 NM/1 NM (ERK1/2) [1]TARGET: ERK1/2SCH772984 IS A NOVEL AND SELECTIVE INHIBITOR 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 50 MG/ML
SCH772984 IS A NOVEL, SPECIFIC INHIBITOR OF ERK1/2 WITH IC50 OF 4 NM AND 1 NM, RESPECTIVELY.IC50 VALUE: 4 NM/1 NM (ERK1/2) [1]TARGET: ERK1/2SCH772984 IS A NOVEL AND SELECTIVE INHIBITOR 1 * 5 mg



