10103 Results for: "ZARGES LEICHTBAU GMBH&"
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
TALTOBULIN (HTI-286 SPA-110) IS AN ANALOGUE OF HEMIASTERLIN POTE NT TUBULIN INHIBITOR ADCS CYTOTOXIN.IC50 VALUE:TARGET: TUBULININ VITRO: HTI-286 SIGNIFICANTLY INHIBITED PROLIFERATIO 1 * 50 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
TALTOBULIN (HTI-286 SPA-110) IS AN ANALOGUE OF HEMIASTERLIN POTE NT TUBULIN INHIBITOR ADCS CYTOTOXIN.IC50 VALUE:TARGET: TUBULININ VITRO: HTI-286 SIGNIFICANTLY INHIBITED PROLIFERATIO 1 * 50 mg
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405 Target Protein,,MPRA Clonality,,Polyclonal Storage/Stability,,-20°C/1 year Application,,WB,IF/ICC,ELISA Recommended Dilution,,WB 1:500~1:1000, IF/ICC 1:100-1:500 Concentration,,1 mg/ml Reactive Species,,Human,Mouse Host Species,,Rabbit Immunogen, 1 * 100 µG
Supplier: G-Biosciences
405 Target Protein,,MPRA Clonality,,Polyclonal Storage/Stability,,-20°C/1 year Application,,WB,IF/ICC,ELISA Recommended Dilution,,WB 1:500~1:1000, IF/ICC 1:100-1:500 Concentration,,1 mg/ml Reactive Species,,Human,Mouse Host Species,,Rabbit Immunogen, 1 * 100 µG
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Target Protein,,P2RY6 Clonality,,Polyclonal Storage/Stability,,-20°C/1 year Application,,WB,ELISA Recommended Dilution,,WB 1:500-2000 ELISA 1:5000-20000 Concentration,,1 mg/ml Reactive Species,,Human,Rat,Mouse Host Species,,Rabbit Immunogen,,Synthesi 1 * 50 µG
Supplier: G-Biosciences
Target Protein,,P2RY6 Clonality,,Polyclonal Storage/Stability,,-20°C/1 year Application,,WB,ELISA Recommended Dilution,,WB 1:500-2000 ELISA 1:5000-20000 Concentration,,1 mg/ml Reactive Species,,Human,Rat,Mouse Host Species,,Rabbit Immunogen,,Synthesi 1 * 50 µG
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 30 MG/ML
RO3280 IS A POTENT, HIGHLY SELECTIVE INHIBITOR OF POLO-LIKE KIN ASE 1 (PLK1) WITH IC50 OF 3 NM.IC50 VALUE: 3 NM (PLK1) [1]TARGET: PLKIN VITRO: DIFLUORO-ANALOG 7 (RO3280) GAVE THE BE 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 30 MG/ML
RO3280 IS A POTENT, HIGHLY SELECTIVE INHIBITOR OF POLO-LIKE KIN ASE 1 (PLK1) WITH IC50 OF 3 NM.IC50 VALUE: 3 NM (PLK1) [1]TARGET: PLKIN VITRO: DIFLUORO-ANALOG 7 (RO3280) GAVE THE BE 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 4.7 MG/ML
FTI-277 HCL IS AN INHIBITOR OF FARNESYL TRANSFERASE (FTASE) A HIGHLY POTENT RAS CAAX PEPTIDOMIMETIC WHICH ANTAGONIZES BOTH H- AND K-RAS ONCOGENIC SIGNALING.IC50 VALUE:TARGET: FTA 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 4.7 MG/ML
FTI-277 HCL IS AN INHIBITOR OF FARNESYL TRANSFERASE (FTASE) A HIGHLY POTENT RAS CAAX PEPTIDOMIMETIC WHICH ANTAGONIZES BOTH H- AND K-RAS ONCOGENIC SIGNALING.IC50 VALUE:TARGET: FTA 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
GENZ-644282 IS A NON-CAMPTOTHECIN INHIBITOR OF TOPOISOMERASE I WIT H POTENTIAL ANTINEOPLASTIC ACTIVITY(IC50=1.2 NM).IC50 VALUE: 1.2 NM [1]TARGET: TOPOISOMERASE IIN VITRO: GENZ-644282 D 1 * 100 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
GENZ-644282 IS A NON-CAMPTOTHECIN INHIBITOR OF TOPOISOMERASE I WIT H POTENTIAL ANTINEOPLASTIC ACTIVITY(IC50=1.2 NM).IC50 VALUE: 1.2 NM [1]TARGET: TOPOISOMERASE IIN VITRO: GENZ-644282 D 1 * 100 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 8 MG/ML (19 MM) WATER <1 MG/ML (<1 MM)
LOVASTATIN IS AN INHIBITOR OF HMG-C OA REDUCTASE WITH IC50 OF 3.4 NM, USED FOR LOWERING CHOLESTEROL (HYPOLIPIDEMIC AGENT). TARGET: HMG-COA REDUCTASELOVAS 1 * 50 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO 8 MG/ML (19 MM) WATER <1 MG/ML (<1 MM)
LOVASTATIN IS AN INHIBITOR OF HMG-C OA REDUCTASE WITH IC50 OF 3.4 NM, USED FOR LOWERING CHOLESTEROL (HYPOLIPIDEMIC AGENT). TARGET: HMG-COA REDUCTASELOVAS 1 * 50 mg
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VarioPrep HPLC column VP 15/50 NUCLEODUR C18 ec length: 15 mm, ID: 50 mm pack of 1 - compatible with VarioPrep HPLC column with ID 50 mm or larger - requires VP guard column holder 50 mm (short version, p/n 718255) 1 * 1 items
Supplier: MACHEREY-NAGEL
VarioPrep HPLC column VP 15/50 NUCLEODUR C18 ec length: 15 mm, ID: 50 mm pack of 1 - compatible with VarioPrep HPLC column with ID 50 mm or larger - requires VP guard column holder 50 mm (short version, p/n 718255) 1 * 1 items
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
KH-CB19 IS A POTENT AND HIGHLY SPECIFIC INHIBITOR OF THE CDC2-LIKE KINASE ISOFORMS 1 AND 4 (CLK1/CLK4).IC50 VALUE: 20 NM (CLK1) [1]TARGET: CLK1/4 INHIBITORIN VITRO: KH-CB19 SHOWED POT 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
KH-CB19 IS A POTENT AND HIGHLY SPECIFIC INHIBITOR OF THE CDC2-LIKE KINASE ISOFORMS 1 AND 4 (CLK1/CLK4).IC50 VALUE: 20 NM (CLK1) [1]TARGET: CLK1/4 INHIBITORIN VITRO: KH-CB19 SHOWED POT 1 * 5 mg
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Target Protein,,MB Clonality,,Polyclonal Storage/Stability,,-20°C/1 year Application,,WB,IHC,IF/ICC,ELISA Recommended Dilution,,WB,,1:500-1:2000 IHC,,1:50-1:200, IF/ICC 1:100-1:500 Concentration,,1 mg/ml Reactive Species,,Human,Mouse,Rat Host Species 1 * 200 µG
Supplier: G-Biosciences
Target Protein,,MB Clonality,,Polyclonal Storage/Stability,,-20°C/1 year Application,,WB,IHC,IF/ICC,ELISA Recommended Dilution,,WB,,1:500-1:2000 IHC,,1:50-1:200, IF/ICC 1:100-1:500 Concentration,,1 mg/ml Reactive Species,,Human,Mouse,Rat Host Species 1 * 200 µG
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 50 MM IN DMSO
GSK126 IS A POTENT, HIGHLY SELECTIVE, S-ADENOSYL-METHIONINE-COMPET ITIVE, SMALL-MOLECULE INHIBITOR OF EZH2 METHYLTRANSFERASE WITH KI VALUE OF 0.5 NM.IC50 VALUE: 0.5 NM (KI)TARGET: EZH2 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 50 MM IN DMSO
GSK126 IS A POTENT, HIGHLY SELECTIVE, S-ADENOSYL-METHIONINE-COMPET ITIVE, SMALL-MOLECULE INHIBITOR OF EZH2 METHYLTRANSFERASE WITH KI VALUE OF 0.5 NM.IC50 VALUE: 0.5 NM (KI)TARGET: EZH2 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 100 MM IN DMSO
IWR-1(IWR-1-ENDO) IS A NOVEL SMALL-MOLECULE INHIBITOR OF WNT SIGN ALING BY STABILIZING THE AXIN DESTRUCTION COMPLEX WITH AN EC50 OF 0.2 UM.IC50 VALUE: 0.2 UM (EC50) [1]TARGET: WNT SIG 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 100 MM IN DMSO
IWR-1(IWR-1-ENDO) IS A NOVEL SMALL-MOLECULE INHIBITOR OF WNT SIGN ALING BY STABILIZING THE AXIN DESTRUCTION COMPLEX WITH AN EC50 OF 0.2 UM.IC50 VALUE: 0.2 UM (EC50) [1]TARGET: WNT SIG 1 * 5 mg
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Antibody Immunotag™ TGF ß Receptor I (ABT-TGFR1) mouse mAb-FITC Target Protein: TGF ß Receptor I (2F2) Clonality: Monoclonal Storage/Stability: -20°C/1 year Concentration: 1 mg/ml Reactive Species: Human Host Species: Mouse Immunogen: Synthesized pep 1 * 100 µG
Supplier: G-Biosciences
Antibody Immunotag™ TGF ß Receptor I (ABT-TGFR1) mouse mAb-FITC Target Protein: TGF ß Receptor I (2F2) Clonality: Monoclonal Storage/Stability: -20°C/1 year Concentration: 1 mg/ml Reactive Species: Human Host Species: Mouse Immunogen: Synthesized pep 1 * 100 µG
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥5MG/ML WATER <1.2MG/ML ETHANOL ≥36MG/ML
CYCLOPAMINE(11-DEOXOJERVINE) IS A SPECIFIC HEDGEHOG (HH) SIGNALING PATHWAY ANTAGONIST OF SMOOTHENED (SMO) WITH IC50 OF 46 NM.IC50 VALUE: 46 NM [1]TARGET 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥5MG/ML WATER <1.2MG/ML ETHANOL ≥36MG/ML
CYCLOPAMINE(11-DEOXOJERVINE) IS A SPECIFIC HEDGEHOG (HH) SIGNALING PATHWAY ANTAGONIST OF SMOOTHENED (SMO) WITH IC50 OF 46 NM.IC50 VALUE: 46 NM [1]TARGET 1 * 5 mg
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Target Protein,,P2RY6 Clonality Polyclonal Application,,WB,ELISA Recommended Dilution,,WB 1:500-2000 ELISA 1:5000-20000 Concentration,,1 mg/ml Reactive Species,,Human,Rat,Mouse Host Species,,Rabbit Immunogen,,Synthesized peptide derived from human pr 1 * 50 µG
Supplier: G-Biosciences
Target Protein,,P2RY6 Clonality Polyclonal Application,,WB,ELISA Recommended Dilution,,WB 1:500-2000 ELISA 1:5000-20000 Concentration,,1 mg/ml Reactive Species,,Human,Rat,Mouse Host Species,,Rabbit Immunogen,,Synthesized peptide derived from human pr 1 * 50 µG
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SOLUBILITY: DMSO 95 MG/ML WATER 95 MG/ML ETHANOL <1 MG/ML
RIGOSERTIB (ON-01910) IS A NON-ATP-COMPETITIVE INHIBITOR OF PLK1 WITH IC50 OF 9 NM SHOWS 30-FOLD GREATER SELECTIVITY AGAINST PLK2 AND NO ACTIVITY TO PLK3.IC50 VALUE: 9 NM [1] TARGET: PL 1 * 5 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: DMSO 95 MG/ML WATER 95 MG/ML ETHANOL <1 MG/ML
RIGOSERTIB (ON-01910) IS A NON-ATP-COMPETITIVE INHIBITOR OF PLK1 WITH IC50 OF 9 NM SHOWS 30-FOLD GREATER SELECTIVITY AGAINST PLK2 AND NO ACTIVITY TO PLK3.IC50 VALUE: 9 NM [1] TARGET: PL 1 * 5 mg
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SOLUBILITY: DMSO: ≥ 30 MG/ML
AZ191 IS A POTENT SMALL MOLECULE INHIBITOR THAT SELECTIVELY INHIBITS DYRK1B WITH IC50 OF 17 NM SELE CTIVE FOR DYRK1B OVER BOTH DYRK1A AND DYRK2.IC50 VALUE: 17 NM [1]TARGET: DYRK1B INHIBITORIN VITRO: USING IN VITRO KIN 1 * 50 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: DMSO: ≥ 30 MG/ML
AZ191 IS A POTENT SMALL MOLECULE INHIBITOR THAT SELECTIVELY INHIBITS DYRK1B WITH IC50 OF 17 NM SELE CTIVE FOR DYRK1B OVER BOTH DYRK1A AND DYRK2.IC50 VALUE: 17 NM [1]TARGET: DYRK1B INHIBITORIN VITRO: USING IN VITRO KIN 1 * 50 mg
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CF™440 maleimide is a bluish green fluorescent dye with a maleimide reactive group, which can be used to label a target molecule wi th a thiol group. CF™440 (abs/em=440 nm/515 nm) is a superior alternative to Alexa Fluor 430 owing to its exceptiona 1 * 1 µmol
Supplier: Biotium
CF™440 maleimide is a bluish green fluorescent dye with a maleimide reactive group, which can be used to label a target molecule wi th a thiol group. CF™440 (abs/em=440 nm/515 nm) is a superior alternative to Alexa Fluor 430 owing to its exceptiona 1 * 1 µmol
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Feuchte/Temperatur-Transmitter EE22 mit abgesetztem Fühler L= 2 Meter Bereich 0..100%rH, -40..80°C, Fühlerlänge ca. 75mm, mit abgese tztem rH/T-Fühler, Kabellänge 2 Meter, Ausgang 4..20mA, Speisung 20-35V DC, Anschlussstecker 4polig (m) Genauigkeit F 1 * 1 Pack.
Supplier: ELPRO-BUCHS
Feuchte/Temperatur-Transmitter EE22 mit abgesetztem Fühler L= 2 Meter Bereich 0..100%rH, -40..80°C, Fühlerlänge ca. 75mm, mit abgese tztem rH/T-Fühler, Kabellänge 2 Meter, Ausgang 4..20mA, Speisung 20-35V DC, Anschlussstecker 4polig (m) Genauigkeit F 1 * 1 Pack.
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥9MG/ML WATER <1.2MG/ML ETHANOL ≥60MG/ML
GSK461364 IS A POTENT SMALL MOLECU LE POLO-LIKE KINASE 1 (PLK1) INHIBITOR WITH A KI OF 2.2 NM. IC50 VALUE: 2.2 NM(KI)TARGET: PLK1IN VITRO: GSK461364 IS 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥9MG/ML WATER <1.2MG/ML ETHANOL ≥60MG/ML
GSK461364 IS A POTENT SMALL MOLECU LE POLO-LIKE KINASE 1 (PLK1) INHIBITOR WITH A KI OF 2.2 NM. IC50 VALUE: 2.2 NM(KI)TARGET: PLK1IN VITRO: GSK461364 IS 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
SIMEPREVIR (TMC 435350) IS A POTENT INHIBITOR OF HCV NS3/4A PROTEA SE (KI = 0.36 NM) AND VIRAL REPLICATION (REPLICON EC50 = 7.8 NM). IC50 VALUE: 0.36 NM(KI) 7.8 NM (EC50) [1]TARGET: H 1 * 1 mL
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
SIMEPREVIR (TMC 435350) IS A POTENT INHIBITOR OF HCV NS3/4A PROTEA SE (KI = 0.36 NM) AND VIRAL REPLICATION (REPLICON EC50 = 7.8 NM). IC50 VALUE: 0.36 NM(KI) 7.8 NM (EC50) [1]TARGET: H 1 * 1 mL
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
JNJ-17203212 IS A NOVEL AND SELECTIVE TRPV1 ANTAGONIST, WITH IC50 OF 65 NM AND 102 NM FOR HUMAN TRPV1 AND RAT TRPV1.IC50 VALUE: 65 NM (HUMAN TRPV1), 102 NM (RAT TRPV1)TARGET: TRPVIN VI 1 * 50 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
JNJ-17203212 IS A NOVEL AND SELECTIVE TRPV1 ANTAGONIST, WITH IC50 OF 65 NM AND 102 NM FOR HUMAN TRPV1 AND RAT TRPV1.IC50 VALUE: 65 NM (HUMAN TRPV1), 102 NM (RAT TRPV1)TARGET: TRPVIN VI 1 * 50 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 51 MG/ML
ABT-199 (GDC-0199) IS A BCL-2-SELECTIVE INHIBITOR WITH KI OF <0 .01 NM, >4800-FOLD MORE SELECTIVE VERSUS BCL-XL AND BCL-W, AND NO ACTIVITY TO MCL-1. IC50 VALUE: <0.01 NM (KI)TARGET: 1 * 100 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 51 MG/ML
ABT-199 (GDC-0199) IS A BCL-2-SELECTIVE INHIBITOR WITH KI OF <0 .01 NM, >4800-FOLD MORE SELECTIVE VERSUS BCL-XL AND BCL-W, AND NO ACTIVITY TO MCL-1. IC50 VALUE: <0.01 NM (KI)TARGET: 1 * 100 mg