"MEDCHEMEXPRESS"
SOLUBILITY: SOLUBLE TO 100 MM IN DMSO AND TO 50 MM IN ETHANOL
CASIN IS A SELECTIVE GTPASE CDC42 INHIBITOR WITH IC50 OF 2 UM. IN V ITRO: TREATMENT WITH CASIN (5 UM) REDUCED THE ELEVATED LEVEL OF ACTIVE CDC42 OBSERVED IN AGED PRIMITIVE HEMATOPOIETIC 1 * 5 mg
Supplier: MEDCHEMEXPRESS
SOLUBILITY: SOLUBLE TO 100 MM IN DMSO AND TO 50 MM IN ETHANOL
CASIN IS A SELECTIVE GTPASE CDC42 INHIBITOR WITH IC50 OF 2 UM. IN V ITRO: TREATMENT WITH CASIN (5 UM) REDUCED THE ELEVATED LEVEL OF ACTIVE CDC42 OBSERVED IN AGED PRIMITIVE HEMATOPOIETIC 1 * 5 mg
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RIGOSERTIB (SODIUM) 1 * 5 mg
Supplier: MEDCHEMEXPRESS
RIGOSERTIB (SODIUM) 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
ML216(CID-49852229) IS A POTENT INHIBITOR OF THE DNA UNWINDING ACT IVITY OF BLM HELICASE SHOWING SIMILAR IC50S OF 3.0 AND 0.97 ΜM FOR FULL LENGTH BLM AND BLM636–1298 RESPECTIVELY.IC50 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
ML216(CID-49852229) IS A POTENT INHIBITOR OF THE DNA UNWINDING ACT IVITY OF BLM HELICASE SHOWING SIMILAR IC50S OF 3.0 AND 0.97 ΜM FOR FULL LENGTH BLM AND BLM636–1298 RESPECTIVELY.IC50 1 * 5 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 100 MM IN DMSO ; 10 MM IN ETHANOL;
CH-223191 IS A LIGAND-SELECTIVE ANTAGONIST OF THE AH (DIOXIN) RECEPTOR.IC50 VALUE: TARGET: AHR ANTAGONISTIN VITRO: CH-223191 PREFERENTIALLY INHIBITS THE ABILITY O 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 100 MM IN DMSO ; 10 MM IN ETHANOL;
CH-223191 IS A LIGAND-SELECTIVE ANTAGONIST OF THE AH (DIOXIN) RECEPTOR.IC50 VALUE: TARGET: AHR ANTAGONISTIN VITRO: CH-223191 PREFERENTIALLY INHIBITS THE ABILITY O 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥42MG/ML WATER <1.2MG/ML ETHANOL <1.2MG/ML
SP600125 IS A BROAD-SPECTRUM JNK INHIBITOR FOR JNK1, JNK2 AND JNK3 WITH IC50 OF 40 NM, 40 NM AND 90 NM, RESPECTIVELY 10-FOLD GREATER SELECTIVITY AGA 1 * 10 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO ≥42MG/ML WATER <1.2MG/ML ETHANOL <1.2MG/ML
SP600125 IS A BROAD-SPECTRUM JNK INHIBITOR FOR JNK1, JNK2 AND JNK3 WITH IC50 OF 40 NM, 40 NM AND 90 NM, RESPECTIVELY 10-FOLD GREATER SELECTIVITY AGA 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 5 MG/ML, H2O: < 4.9 MG/ML
UNC2025 IS A POTENT AND ORALLY BIOAVAILABLE ME R/FLT3 DUAL INHIBITOR WITH IC50 OF 0.8/0.74 NM FOR MER/FLT3.IC50 VALUE: 0.8/0.74 NM(MER/FLT3)TARGET: MER/FLT3 INHIBIT 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO: ≥ 5 MG/ML, H2O: < 4.9 MG/ML
UNC2025 IS A POTENT AND ORALLY BIOAVAILABLE ME R/FLT3 DUAL INHIBITOR WITH IC50 OF 0.8/0.74 NM FOR MER/FLT3.IC50 VALUE: 0.8/0.74 NM(MER/FLT3)TARGET: MER/FLT3 INHIBIT 1 * 5 mg
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VINORELBINE [71486-22-1] 1 * 10 mg
Supplier: MEDCHEMEXPRESS
VINORELBINE [71486-22-1] 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
PF-3758309 IS AN INHBITOR OF PAKS WITH IC50 OF 1.3 NM FOR PAK4 IN HBITS TUMOR GROWTH IN HCT116, A549, M24MET AND OTHER XENOGRAFT TUMOR MODELS..IC50 VALUE: 1.3 NM (PAK4)TARGET: PAKSIN 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: 10 MM IN DMSO
PF-3758309 IS AN INHBITOR OF PAKS WITH IC50 OF 1.3 NM FOR PAK4 IN HBITS TUMOR GROWTH IN HCT116, A549, M24MET AND OTHER XENOGRAFT TUMOR MODELS..IC50 VALUE: 1.3 NM (PAK4)TARGET: PAKSIN 1 * 5 mg
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KU-60019 [925701-46-8] 1 * 10 mg
Supplier: MEDCHEMEXPRESS
KU-60019 [925701-46-8] 1 * 10 mg
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LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO:36MG/ML
AZD3965 IS A SELECTIVE INHIBITOR OF MONOCARBOXYLATE TRANSPORTER 1 ( MCT1) WITH A BINDING AFFINITY OF 1.6 NM, IS 6 FOLD SELECTIVE OVER MCT2 AND DOES NOT INHIBIT MCT4 AT 10 ΜM.IC50 VALUE: 1 * 5 mg
Supplier: MEDCHEMEXPRESS
LIQUID FORMAT IS 10MM*1ML IN DMSO
SOLUBILITY: DMSO:36MG/ML
AZD3965 IS A SELECTIVE INHIBITOR OF MONOCARBOXYLATE TRANSPORTER 1 ( MCT1) WITH A BINDING AFFINITY OF 1.6 NM, IS 6 FOLD SELECTIVE OVER MCT2 AND DOES NOT INHIBIT MCT4 AT 10 ΜM.IC50 VALUE: 1 * 5 mg
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SOLUBILITY: DMSO: ≥ 33 MG/ML
BI605906, A NOVEL INHIBITOR OF IKKΒ, INHIBITS IKKΒ WITH AN IC50 VALUE OF 380 NM WHEN ASSAYED AT 0.1 MM ATP. IC50 VALUE: 380 NMTARGET: IKKΒIN VITRO: BI605906 IS A NOVEL PHARMACOLOGICAL INHIBITORS OF THE IKK FAMILY, INHI 1 * 1 mL
Supplier: MEDCHEMEXPRESS
SOLUBILITY: DMSO: ≥ 33 MG/ML
BI605906, A NOVEL INHIBITOR OF IKKΒ, INHIBITS IKKΒ WITH AN IC50 VALUE OF 380 NM WHEN ASSAYED AT 0.1 MM ATP. IC50 VALUE: 380 NMTARGET: IKKΒIN VITRO: BI605906 IS A NOVEL PHARMACOLOGICAL INHIBITORS OF THE IKK FAMILY, INHI 1 * 1 mL
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[EN]GILTERITINIB 1 * 50 mg
Supplier: MEDCHEMEXPRESS
[EN]GILTERITINIB 1 * 50 mg
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