Order Entry
Belgium
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CinnGEL 2-methylester
CinnGEL 2-methylester
  ENZOBMLPR1150001
 :  
undefined
CinnGEL 2-methylester
  ENZOBMLPR1150001
 :  

 

  • Pk:
    1 mg
  • Seq:
    02
  • Protein/peptide name:
    CinnGEL 2-methylester

 

 

PTP1B inhibitor

Novel peptoid inhibitor of PTP1B (IC50=1,3 µM). Methyl ester (for cell permeability) is hydrolyzed to active inhibitor by intracellular esterases.